Synthesis of novel N-protected hydrophobic phenylalanines and their application in potential antibacterials.

نویسندگان

  • Timothy P Boyle
  • John B Bremner
  • Jonathan A Coates
  • John Deadman
  • Paul A Keller
  • Stephen G Pyne
  • Kittiya Somphol
چکیده

An efficient synthesis of two new N-acetyl-4'-arylphenylalanines is described together with their incorporation into a number of cationic peptoid antibacterial agents, one of which had an MIC of 7.8 microg/mL against Staphylococcus aureus.

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عنوان ژورنال:
  • European journal of medicinal chemistry

دوره 44 3  شماره 

صفحات  -

تاریخ انتشار 2009