Synthesis of novel N-protected hydrophobic phenylalanines and their application in potential antibacterials.
نویسندگان
چکیده
An efficient synthesis of two new N-acetyl-4'-arylphenylalanines is described together with their incorporation into a number of cationic peptoid antibacterial agents, one of which had an MIC of 7.8 microg/mL against Staphylococcus aureus.
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ورودعنوان ژورنال:
- European journal of medicinal chemistry
دوره 44 3 شماره
صفحات -
تاریخ انتشار 2009